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Serotonin Antagonists

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Definition: Drugs that bind to but do not activate serotonin receptors, thereby blocking the actions of serotonin or SEROTONIN RECEPTOR AGONISTS.  GEN or unspecified; prefer specifics; differentiate from SEROTONIN UPTAKE INHIBITORS: read MeSH definition; do not confuse with SEROTONIN AGONISTS; DF: SEROTONIN ANTAG   
See Also Serotonin Uptake Inhibitors
Examples Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists 		Other names Serotonin Blockaders; Antiserotonergic Agents; 5-Hydroxytryptamine Antagonists; 5-HT Antagonists; Blockaders, Serotonin; Antagonists, 5 Hydroxytryptamine; Antagonists, 5 HT; Agents, Antiserotonergic; 5 Hydroxytryptamine Antagonists; 5 HT Antagonists; Antagonists, Serotonin; Antagonists, 5-Hydroxytryptamine; Antagonists, 5-HT
Substances having this pharmacologic action: clovoxamine; cianopramine; 6-nitroquipazine; CQ 32085; LY 53857; bemesetron; tolfenamic acid; pipamperone; wortmannin; iprazochrome; xylamidine; GR 127935; alosetron; EEDQ; Pindolol; Pizotyline; Cinanserin; Nafronyl; Ritanserin; Ondansetron; Granisetron; Risperidone; Fenclonine; Lysergic Acid Diethylamide; Metergoline; Methiothepin; Methysergide; N,N-Dimethyltryptamine; Clozapine; Bufotenin; Cyproheptadine; Mianserin; Ketanserin; ziprasidone; SB 206553; DuP 734; MDL 100907; WAY 100135; GR 113808; palonosetron; dotarizine; SB 204070A; 4-(2'-methoxyphenyl)-1-(2'-(N-(2''-pyridinyl)-4-iodobenzamido)ethyl)piperazine; WAY 100635; azasetron; fananserin; ramosetron; SDZ 205-557; SR 46349B; dolasetron mesylate; deramciclane; binospirone mesylate; UH 301; sarpogrelate; zatosetron; 2-((2-(dimethylamino)ethyl)thio)-3-phenylquinoline; zacopride; McN 5652; 1-(2-methoxyphenyl)-4-(4-(2-phthalimido)butyl)piperazine; cyanopindolol; amperozide; renzapride; setoperone; tropisetron
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-2,2-diphenylcyclopentan-1-ol  0   *Cyclopentanes *Piperazines Serotonin Antagonists Receptor, Serotonin, 5-HT1A. J Med Chem. 2012 Jan 12;55(1):23-36.
((5,5-diphenyloxolan-2-yl)methyl)(2-phenoxyethyl)amine  0   *Furans Serotonin Antagonists Receptor, Serotonin, 5-HT1A. J Med Chem. 2012 Jan 12;55(1):23-36.
CMP Y compound  0   *Guanidines *Sulfonamides Serotonin Antagonists. Neurobiol Learn Mem. 2011 Sep;96(2):392-402.
CMP X compound  0   *Guanidines *Sulfonamides Serotonin Antagonists. Neurobiol Learn Mem. 2011 Sep;96(2):392-402.
(2-(6-fluoro-1H-indol-3-yl)-ethyl)-(3-(2,2,3,3-tetrafluoropropoxy)benzyl)amine  0   *Benzylamines *Indoles Serotonin Antagonists. Int J Neuropsychopharmacol. 2010 Sep;13(8):1021-33.
MDL 28727  0   Organic Chemicals Serotonin Antagonists. Synapse 1994 Jul;17(3):173-81
GR 65630  117186-80-8   *Imidazoles *Indoles Serotonin Antagonists Receptors, Serotonin, 5-HT3. Neurosci Lett 1988;94(1-2):156
CGS 1068B  114470-88-1   Organic Chemicals Serotonin Antagonists. Physiol Behav 1988;42(4):319

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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012
Warning: the drugs or drug combinations referred to here may be similar or related, but are not be the same ones and may not have the same pharmacological action as other substances described on the same page or in the same row. Please refer to product monograph or to your doctor
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