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Cyproheptadine
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Definition
: A serotonin antagonist and a histamine H1 blocker used as antipruritic, appetite stimulant, antiallergic, and for the post-gastrectomy dumping syndrome, etc.
a histamine H1 antag & serotonin antag
Pharmacological Action
Anti-Allergic Agents
;
Antipruritics
;
Gastrointestinal Agents
;
Histamine H1 Antagonists
;
Serotonin Antagonists
Examples
Loratadine
Other names
Viternum; Peritol; Periactin; Dihexazin; Antergan
Drugs
*
:
CYPROHEPTADINE HYDROCHLORIDE
;
PERIACTIN
Substance
CAS Registry & name
Categories
Source
Drugs
*
rupatadine
156611-76-6
Cyproheptadine/*analogs & derivatives
Platelet Activating Factor/antagonists & inhibitors.
J Pharmacol Exp Ther 1997 Jan;280(1):114-21
desmethylcyproheptadine 10,11-
epoxide
54191-03-6
Cyproheptadine/*analogs & derivatives.
Cell Biol Toxicol 1989;5(2):129
cyproheptadine 10,11-
epoxide
54191-04-7
Cyproheptadine/*analogs & derivatives.
Cell Biol Toxicol 1989;5(2):129
3-
methoxycyproheptadine
77263-46-8
Cyproheptadine/*analogs & derivatives.
J Pharmacol Exp Ther 1988;247(2):796
Sch 399
98125-69-0
*Dextromethorphan
*Pseudoephedrine
Cyproheptadine/*analogs & derivatives
Drug Combinations.
Clin Ther 1984;6(4):475
azatadine maleate, pseudoephedrine sulfate drug combination
0
*Pseudoephedrine
Cyproheptadine/*analogs & derivatives
Drug Combinations.
Pharma Action
Histamine H1 Antagonists
;
Sympathomimetics
Pharmatherapeutica 1984;3(10):657
L 646462
89149-85-9 5H-
Dibenzo(a,d)cycloheptene-
3-
carboxylic acid, 5-
(1-
methyl-
4-
piperidinylidene)-
, (3-
methyl-
2,5-
dioxo-
1-
imidazolidinyl)methyl ester, (-
)
Cyproheptadine/*analogs & derivatives.
J Pharmacol Exp Ther 1984;229(3):775
desmethylcyproheptadine
14051-46-8
Cyproheptadine/*analogs & derivatives.
J Endocrinol 1983;96(3):395
MK 711
63141-67-3
Cyproheptadine/*analogs & derivatives
Appetite/drug effects.
Drug Metab Dispos 1981;9(5):428
cyproheptadine glucuronide
66167-97-3 Piperidinium, 4-
(5H-
dibenzo(a,d)cyclohepten-
5-
ylidene)-
1-
beta-
D-
glucopyranuronosyl-
1-
methyl
Cyproheptadine/*analogs & derivatives.
Drug Metab Dispos 1980;8(6):422
cyproheptadinium methiodide
74927-10-9
Cyproheptadine/*analogs & derivatives.
J Med Chem 1980;23(11):1255
1-
cyclopropylmethyl-
4-
(3-
trifluoromethylthio-
5H-
dibenzo(a,d)cyclohepten-
5-
ylidene)piperidine
0
Cyproheptadine/*analogs & derivatives.
J Med Chem 20(8):1013;1977
azatadine
3964-81-6 6,11-
dihydro-
11-
(1-
methyl-
4-
piperidylidene)-
5H-
benzo(5,6)cyclohepta(1,2-
b)pyridine
Cyproheptadine/*analogs & derivatives.
Pharma Action
Histamine H1 Antagonists
Agents Actions 4(4):264;1974; J Lab Clin Med 90(4):638;1977; Med Lett 19(19):77;1977; Radioisotopes 26(1):33;1977
TRINALIN
;
OPTIMINE