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ψ
ψ
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Telomerase
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Definition
: An essential ribonucleoprotein reverse transcriptase that adds telomeric DNA to the ends of eukaryotic CHROMOSOMES.
See Also
Telomere Homeostasis
Other names
Transcriptase, Telomerase Reverse; Subunit, Telomerase Catalytic; Reverse Transcriptase, Telomerase; Catalytic Subunit, Telomerase; Telomerase Reverse Transcriptase Catalytic Subunit; Telomerase Reverse Transcriptase; Telomerase Catalytic Subunit
Substance
CAS Registry & name
Categories
Source
Drugs
*
EST1 protein, S pombe
EC 2.7.7.49
*Telomerase
*Schizosaccharomyces pombe Proteins
Protein Subunits.
Nat Struct Mol Biol. 2011 Dec;18(12):1408-13
2,2'-
(1,3-
phenylene)-
bis-
(5-
(4-
(2-
hydroxyethyl)-
1-
piperazinyl)-
1H-
benzimidazole)
0
*Benzimidazoles
*Piperazines
Telomerase/antagonists & inhibitors.
Bioconjug Chem 2010 Jul 21;21(7):1148-59
2,2'-
(1,4-
phenylene)-
bis-
(5-
(4-
(2-
hydroxyethyl)-
1-
piperazinyl)-
1H-
benzimidazole)
0
*Benzimidazoles
*Piperazines
Telomerase/antagonists & inhibitors.
Bioconjug Chem 2010 Jul 21;21(7):1148-59
5'-
oleic-
TAGGGTTAGACAA-
3'
0
*Oligonucleotides
Telomerase/antagonists & inhibitors.
Breast Cancer Res Treat 20-09 Nov;118(1):21-32
telomerase Cajal body protein 1, human
EC 2.7.7.49
*Telomerase.
Science. 2009 Jan 30;323(5914):644-8
TERT protein, Arabidopsis
EC 2.7.7.49
*Telomerase
*Arabidopsis Proteins
Protein Subunits.
FEBS Lett 1999 Sep 3;457(3):465-9
hTERT mp30-
38 peptide
EC 2.7.7.-
*Telomerase
Peptide Fragments.
Cancer Immunol Immunother 2007 Nov;56(11):1755-63
telomerase reverse transcriptase p572Y, human
EC 2.7.7.49
*Telomerase.
J Clin Oncol 2007 Jul 1;25(19):2727-34
N'-
(10H-
indolo(3,2-
b)quinolin-
11-
yl)-
N,N-
dimethylpropane-
1,3-
diamine
0
*Diamines
*Quinolines
Telomerase/antagonists & inhibitors.
Leukemia 2007 Jun;21(6):1300-2
GV1001 peptide
EC 2.7.7.-
*Peptide Fragments
*Telomerase.
Cancer Immunol Immunother 2006 Dec;55(12):1553-64
SMG6 protein, human
EC 2.7.7.49
*Telomerase
Protein Subunits.
Curr Biol 2003 Apr 1;13(7):568-74
chrolactomycin
0
*Diterpenes
Telomerase/antagonists & inhibitors.
Curr Biol 2006 Feb;13(2):183-90
trt1 protein, S pombe
0
*Telomerase
*Schizosaccharomyces pombe Proteins.
Tert protein, mouse
EC 2.7.7.49
*Telomerase.
TERT protein, human
EC 2.7.7.49
*Telomerase.
EST2 protein, S cerevisiae
EC 2.7.7.49
*Telomerase
*Saccharomyces cerevisiae Proteins.
PIF1 protein, human
EC 5.99.-
*DNA Helicases
Telomerase/antagonists & inhibitors.
Nucleic Acids Res 2006;34(5):1393-404
GRN163L peptide
0
*Oligonucleotides
Telomerase.
Hepatology 2005 Nov;42(5):1127-36
Zap3 protein, mouse
0
*Nucleoproteins
Telomerase/antagonists & inhibitors.
Mech Dev 2004 Dec;121(12):1509-22
EST3 protein, S cerevisiae
EC 2.7.7.49
*Telomerase
*Saccharomyces cerevisiae Proteins.
2,6-
bis(3-
(N-
piperidino)propionamido)anthracene-
9,10-
dione
0
*Anthraquinones
*Piperidines
Telomerase/antagonists & inhibitors.
Gastroenterology 2004 May;126(5):1337-46
BIBR 1532
0
*Aminobenzoic Acids
*Naphthalenes
Telomerase/antagonists & inhibitors.
EMBO J. 2001 Dec 17;20(24):6958-68; J Biol Chem 2002 May 3;277(18):15566-72
BisA compound
0
*Acridines
*Bridged Compounds
Telomerase/antagonists & inhibitors.
J Biomol Struct Dyn 2001 Dec;19(3):505-13
6-
thio-
7-
deaza-
2'-
deoxyguanosine 5'-
triphosphate
0
*Deoxyguanine Nucleotides
Telomerase/antagonists & inhibitors.
Bioorg Chem 2001 Feb;29(1):36-55
PINX1 protein, human
0
*Tumor Suppressor Proteins
Telomerase/antagonists & inhibitors.
Cell 2001 Nov 2;107(3):347-59
3,11-
difluoro-
6,8,13-
trimethyl-
8H-
quino(4,3,2-
kl)acridinium
0
*Acridines
Telomerase/antagonists & inhibitors.
Mol Pharmacol 2001 Nov;60(5):981-8
telomerase reverse transcriptase (540-
548)
EC 2.7.7.-
*Peptide Fragments
*Telomerase.
Eur J Immunol 2001 Sep;31(9):2642-51
telomestatin
0
*Oxazoles
Telomerase.
J Am Chem Soc 2001 Feb 14;123(6):1262-3
telomerase RNA
0
*RNA
*Telomerase.
Gene 1998 Oct 9;221(1):51-58; J Biol Chem 2001 Feb 23;276(8):5856-65
p95 protein, Tetrahymena
0
*RNA-Binding Proteins
*Telomere-Binding Proteins
Telomerase.
Cell 1995 Jun 2;81(5):677-86
FSU oligonucleotide
0
*Oligonucleotides
Telomerase/antagonists & inhibitors.
Anal Biochem 2000 Jun 15;282(1):80-8
protelomerase protein, Bacteriophage N15
EC 2.7.7.-
*Enzyme Precursors
*Viral Proteins
*Telomerase.
Proc Natl Acad Sci U S A 2000 Jul 5;97(14):7721-6
2-
(3-
(trifluoromethyl)phenyl)-
isothiazolin-
3-
one
0
*Thiazoles
Telomerase/antagonists & inhibitors.
Biochemistry 1999 Aug 31;38(35):11501-7
diazaphilonic acid
0
*Benzopyrans
*Carboxylic Acids
Telomerase.
J Antibiotic (Tokyo) 1999 Apr;52(4):412-4
alterperylenol
0
Perylene/*analogs & derivatives
Telomerase/antagonists & inhibitors.
Oncol Res 1998;10(8):449-53
N,N'-
bis(2-
1(piperidino)-
ethyl)-
3,4,9,10-
perylene-
tetracarboxylic diimide
0
*Piperidines
Perylene/*analogs & derivatives
Telomerase/antagonists & inhibitors.
Nat Med 1998 Dec;4(12):1366-7
hTR RNA
0
*Telomerase
*RNA, Untranslated.
Curr Biol 1998 Jan 29;8(3):177-80
TEP1 protein, human
0
*Carrier Proteins
Telomerase
Vault Ribonucleoprotein Particles.
Science 1997 Feb 14;275(5302):973-7
EST1 protein, S cerevisiae
EC 2.7.7.49
*Telomerase
*Saccharomyces cerevisiae Proteins.
Cell 1989 May 19;57(4):633-43
gamma-
rubromycin
27267-71-6 Spiro(benzo(1,2-
b:5,4-
c')dipyran-
2(3H),2'(3'H)-
naphtho(2,3-
b)furan)-
7-
carboxylic acid, 4,5',8',9-
tetrahydro-
4',9',10-
trihydroxy-
7'-
methoxy-
5',8',9-
trioxo-
, methyl ester
*Quinones
Telomerase/antagonists & inhibitors.
Mol Pharmacol 1990;38(1):20
beta-
rubromycin
27267-70-5 Spiro(benzo(1,2-
b:5,4-
c')dipyran-
2(3H),2'(3'H)-
naphtho(1,2-
b)furan)-
7-
carboxylic acid, 4,4',5',9-
tetrahydro-
6',10-
dihydroxy-
7',9'-
dimethoxy-
4',5',9-
trioxo-
, methyl ester
*Quinones
Telomerase/antagonists & inhibitors.
Mol Pharmacol 1990;38(1):20
alpha-
rubromycin
27267-69-2 1H-
2-
Benzopyran-
3-
carboxylic acid, 6-
(2-
(4,9-
dihydro-
8-
hydroxy-
5,7-
dimethoxy-
4,9-
dioxonaphtho(2,3-
b)furan-
2-
yl)ethyl)-
7,8-
dihydroxy-
1-
oxo-
, methyl ester
*Quinones
Telomerase/antagonists & inhibitors.
Mol Pharmacol 1990;38(1);20
tetra(4-
N-
methylpyridyl)porphine
38673-65-3 (4,4',4'',4'''-
(21H,23H)-
porphine-
5,10,15,20-
tetrayl)tetrakis(1-
methylpyridinium)
*Porphyrins
Telomerase/antagonists & inhibitors.
Pharma Action
Anti-Infective Agents
;
Enzyme Inhibitors
;
Photosensitizing Agents
;
Angiogenesis Inhibitors
Nucleic Acids Res 6(9):3093;1979