ψ
| Drug Resistance, Multiple |
| Simultaneous resistance to several structurally and functionally distinct drugs.
| DRUG RESISTANCE, MULTIPLE, BACTERIAL; DRUG RESISTANCE, MULTIPLE, VIRAL; and DRUG RESISTANCE, MULTIPLE, FUNGAL are also available
See Also Genes, MDR; Multidrug Resistance-Associated Proteins; P-Glycoproteins | Other names Multidrug Resistance; Resistance, Multiple Drug; Multiple Drug Resistance; Multi-Drug Resistance; Multidrug Resistance
| |
| Substance | CAS Registry & name | Categories | Source
|
multidrug resistance-associated protein 1
| 0
|
Drug Resistance, Multiple *Multidrug Resistance-Associated Proteins.
|
|
| ABCG2 protein, human
| 0
|
*Neoplasm Proteins *ATP-Binding Cassette Transporters Drug Resistance, Multiple.
|
Biochem Pharmacol. 2005 Jun 23; Proc Natl Acad Sci U S A 1998 Dec 22;95(26):15665-70
|
| multidrug resistance protein 3
| 0
|
*P-Glycoproteins *ATP-Binding Cassette Transporters Drug Resistance, Multiple.
|
Hematol Oncol Clin North Am 1995 Apr;9(2):239-49
|
| valspodar
| 121584-18-7
|
*Cyclosporins Drug Resistance, Multiple P-Glycoprotein.
|
Cancer Res 1991;51(16):4226
|
| major vault protein
| 0
|
*Vault Ribonucleoprotein Particles Drug Resistance, Multiple.
|
Gene 1994 Dec 30;151(1-2):257-60
|
multidrug resistance-associated protein 2
| 0
|
*Membrane Transport Proteins *Multidrug Resistance-Associated Proteins Jaundice, Chronic Idiopathic Drug Resistance, Multiple.
|
Mol Pharmacol 1999 May;55(5):929-37
|
multidrug resistance-associated protein 3
| 0
|
*Multidrug Resistance-Associated Proteins Drug Resistance, Multiple.
|
FEBS Lett 1998 Aug 14;433(1-2):149-52
|
| GF 120918
| 143664-11-3
|
*Acridines *Tetrahydroisoquinolines Drug Resistance, Multiple.
|
Cancer Res 1993 Oct 1;53(19):4595-602
|
| MexB protein, Pseudomonas aeruginosa
| 0
|
*Bacterial Outer Membrane Proteins *Membrane Transport Proteins Drug Resistance, Multiple.
|
J Bacteriol 1993 Nov;175(22):7363-72
|
| MexA protein, Pseudomonas aeruginosa
| 0
|
*Bacterial Outer Membrane Proteins *Membrane Transport Proteins Drug Resistance, Multiple.
|
J Bacteriol 1993 Nov;175(22):7363-72
|
| ABCC5 protein, human
| 0
|
*Multidrug Resistance-Associated Proteins Drug Resistance, Multiple.
|
Cancer Res 1997 Aug 15;57(16):3537-47
|
| zosuquidar trihydrochloride
| 0
|
*Dibenzocycloheptenes *Quinolines Drug Resistance, Multiple.
|
Anticancer Res 1995 May-Jun;15(3):811-4
|
| LmrA protein, Lactococcus lactis
| 0
|
*Bacterial Proteins *Multidrug Resistance-Associated Proteins Drug Resistance, Multiple.
|
Proc Natl Acad Sci U S A 1996 Oct 1;93(20):10668-72
|
| tariquidar
| 206873-63-4
|
*Quinolines Drug Resistance, Multiple.
|
Br J Pharmacol 1999 Sep;128(2):403-11
|
| MexXY protein, Pseudomonas aeruginosa
| 0
|
*Bacterial Proteins Drug Resistance, Multiple.
|
Antimicrob Agents Chemother 1999 Nov;43(11):2624-8
|
| VX 710
| 0
|
*Piperidines *Pyridines Drug Resistance, Multiple.
|
Anticancer Drugs 1997 Feb;8(2):125-40
|
| BmrR protein, bacteria
| 0
|
*Bacterial Proteins *Trans-Activators DNA-Binding Proteins Drug Resistance, Microbial Drug Resistance, Multiple.
|
J Biol Chem 1994 Nov 11;269(45):28506-13
|
| Abcc4 protein, rat
| 0
|
Drug Resistance, Multiple *Multidrug Resistance-Associated Proteins.
|
|
OC 144-093
| 0
|
Drug Resistance, Multiple *Imidazoles.
|
Cancer Res 2000 Jun 1;60(11):2964-72
|
| Abcc5 protein, rat
| 0
|
Drug Resistance, Multiple *Multidrug Resistance-Associated Proteins.
|
|
| QacB protein, Staphylococcus aureus
| 0
|
*Bacterial Proteins *Membrane Transport Proteins Drug Resistance, Multiple.
|
Proc Natl Acad Sci U S A 1996 Apr 16;93(8):3630-5
|
| Abcc5 protein, mouse
| 0
|
Drug Resistance, Multiple *Multidrug Resistance-Associated Proteins.
|
|
| ATPGP1 protein, Arabidopsis
| 0
|
*ATP-Binding Cassette Transporters *Arabidopsis Proteins Drug Resistance, Multiple.
|
Methods Enzymol 1998;292:162-73
|
| HIPK3 protein, human
| EC 2.7.11.1
|
*Protein-Serine-Threonine Kinases *Intracellular Signaling Peptides and Proteins Drug Resistance, Multiple.
|
Gene 1997 Oct 24;200(1-2):35-43; J Biol Chem 1998 Oct 2;273(40):25875-9
|
| hapalosin
| 159542-04-8
|
*Lactams *Lactones *Depsipeptides Drug Resistance, Multiple.
|
J Med Chem 1998 Mar 12;41(6):981-7
|
| R 101933
| 0
|
Drug Resistance, Multiple P-Glycoprotein/antagonists & inhibitors *Benzazepines *Quinolines.
|
Clin Cancer Res 2000 Apr;6(4):1365-71
|
| AadB protein, Acinetobacter sp. SUN
| 0
|
*Bacterial Proteins Drug Resistance, Multiple.
|
FEMS Microbiol Lett 1997 Aug 15;153(2):321-6
|
| RamA protein, Klebsiella
| 0
|
*Bacterial Proteins Drug Resistance, Multiple.
|
Microbiology 1995 Aug;141( Pt 8):1909-20
|
| LfrA protein, Mycobacterium smegmatis
| 0
|
*Bacterial Proteins *Antiporters Drug Resistance, Multiple.
|
Proc Natl Acad Sci U S A 1996 Jan 9;93(1):362-6
|
| Tap protein, Mycobacterium
| 0
|
*Bacterial Proteins *Membrane Transport Proteins Drug Resistance, Microbial Drug Resistance, Multiple.
|
J Bacteriol 1998 Nov;180(22):5836-43
|
| MEF1 protein, human
| 0
|
*DNA-Binding Proteins *Transcription Factors Drug Resistance, Multiple Genes, MDR.
|
Biochemistry 2000 Jan 11;39(1):194-204
|
| RAB6C protein, human
| EC 3.6.1.-
|
Drug Resistance, Multiple *rab GTP-Binding Proteins.
|
Gene 2000 Oct 17;257(1):67-75
|
| FLU1 protein, Candida albicans
| 0
|
*Fungal Proteins *Drug Resistance, Multiple *ATP-Binding Cassette Transporters.
|
Microbiology 2000 Nov;146 ( Pt 11):2743-54
|
| TtgI protein, Pseudomonas putida
| 0
|
Drug Resistance, Multiple *Bacterial Proteins *Membrane Transport Proteins.
|
J Bacteriol 2001 Jul;183(13):3967-73
|
| ATMRP5 protein, Arabidopsis
| 0
|
Drug Resistance, Multiple *Multidrug Resistance-Associated Proteins *Arabidopsis Proteins.
|
|
| VA 033
| 0
|
*Vinca Alkaloids Drug Resistance, Multiple.
|
Eur J Pharmacol 1997 May 30;327(2-3):239-46
|
| MDR1 protein, Filobasidiella neoformans
| 0
|
*Fungal Proteins *ATP-Binding Cassette Transporters Cryptococcus neoformans Drug Resistance, Multiple.
|
Gene 1997 Nov 12;201(1-2):21-9
|
| Pmr1 protein, bacteria
| 0
|
*Bacterial Proteins *ATP-Binding Cassette Transporters Drug Resistance, Multiple.
|
Appl Environ Microbiol 1998 Oct;64(10):3983-8
|
| B 4121
| 0
|
Clofazimine/*analogs & derivatives Drug Resistance, Multiple.
|
Oncol Rep 2000 Jan-Feb;7(1):193-5
|
4-deacetoxyagosterol
| 0
|
Drug Resistance, Multiple *Sterols.
|
Bioorg Med Chem Lett 2000 Nov 20;10(22):2521-4
|
| qacH protein, Staphylococcus saprophyticus
| 0
|
*Bacterial Proteins *Membrane Transport Proteins Drug Resistance, Multiple.
|
FEMS Microbiol Lett 1998 Jan 1;163(1):49-56
|
| FNX1 protein, S pombe
| 0
|
*Drug Resistance, Multiple *Schizosaccharomyces pombe Proteins.
|
Mol Cell Biol 1998 Sep;18(9):5239-46
|
| ATPGP2 protein, Arabidopsis
| 0
|
*ATP-Binding Cassette Transporters *Arabidopsis Proteins Drug Resistance, Multiple.
|
Methods Enzymol 1998;292:162-73
|
GP-88, propafenone-type MDR-modulator
| 0
|
*Phenyl Ethers *Propanols Drug Resistance, Multiple.
|
Bioorg Med Chem Lett 1998 Apr 7;8(7):829-32
|
| MM 36
| 0
|
*Anisoles *Nitriles Drug Resistance, Multiple Drug Resistance, Neoplasm.
|
J Med Chem 1999 May 20;42(10):1687-97
|
| reversin 121
| 0
|
*Oligopeptides Drug Resistance, Multiple.
|
Biochem Pharmacol 1999 Aug 15;58(4):571-86
|
| reversin 205
| 0
|
*Oligopeptides Drug Resistance, Multiple.
|
Biochem Pharmacol 1999 Aug 15;58(4):571-86
|
6-((2-aminoethyl)amino)-2-(2-(dimethylamino)ethyl)-2,3-dihydro-1H,7H-pyrimido(5,6,1-de)acridine-1,3,7-trione
| 0
|
*Acridines *Pyrimidinones Drug Resistance, Multiple Drug Resistance, Neoplasm.
|
J Med Chem 1999 Jul 15;42(14):2535-41
|
9-amino-2-(2-(dimethylamino)ethyl)-6-((2-(dimethylamino)ethyl)amino)-2,3-dihydro-1H,7H-pyrimido(5,6,1-de)acridine-1,3,7-trione
| 0
|
*Acridines *Pyrimidinones Drug Resistance, Multiple Drug Resistance, Neoplasm.
|
J Med Chem 1999 Jul 15;42(14):2535-41
|
9-hydroxy-2-(2-(dimethylamino)ethyl)-6-((2-(dimethylamino)ethyl)amino)-2,3-dihydro-1H,7H-pyrimido(5,6,1-de)acridine-1,3,7-trione
| 0
|
*Acridines *Pyrimidinones Drug Resistance, Multiple Drug Resistance, Neoplasm.
|
J Med Chem 1999 Jul 15;42(14):2535-41
|
| LY 329146
| 0
|
*Sulfonamides *Thiophenes Drug Resistance, Multiple.
|
Bioorg Med Chem Lett 1999 Dec 6;9(23):3381-6
|
| CP 162398
| 0
|
*Piperazines *Quinolines Drug Resistance, Multiple P-Glycoprotein/antagonists & inhibitors.
|
Biochemistry 2000 Jan 11;39(1):75-85
|
| CP 172732
| 0
|
*Piperazines *Thiazoles Drug Resistance, Multiple P-Glycoprotein/antagonists & inhibitors.
|
Biochemistry 2000 Jan 11;39(1):75-85
|
| CP 147673
| 0
|
*Piperazines Drug Resistance, Multiple P-Glycoprotein/antagonists & inhibitors.
|
Biochemistry 2000 Jan 11;39(1):75-85
|
doxorubicin-gallium-transferrin conjugate
| 0
|
Gallium Drug Resistance, Multiple *Doxorubicin *Organometallic Compounds *Transferrin.
|
Anticancer Res 2000 Mar-Apr;20(2A):799-808
|
7-O-benzoylpyripyropene A
| 0
|
Drug Resistance, Multiple *Pyridones *Sesquiterpenes.
|
J Antibiot (Tokyo) 2000 Oct;53(10):1201-6
|
| POHL protein, marine sponge
| 0
|
Drug Resistance, Multiple *Trans-Activators.
|
Environ Toxicol Chem 2001 Jan;20(1):198-204
|
| ArpA protein, Pseudomonas putida
| 0
|
Drug Resistance, Multiple *Bacterial Proteins *Carrier Proteins.
|
Microbiology 2001 Jan;147(Pt 1):43-51
|
| ArpB protein, Pseudomonas putida
| 0
|
Drug Resistance, Multiple *Bacterial Proteins *Membrane Transport Proteins.
|
Microbiology 2001 Jan;147(Pt 1):43-51
|
| ArpC protein, Pseudomonas putida
| 0
|
Drug Resistance, Multiple *Bacterial Proteins *Membrane Transport Proteins.
|
Microbiology 2001 Jan;147(Pt 1):43-51
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