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Calcium Channel Blockers 
A class of drugs that act by selective inhibition of calcium influx through cell membranes or on the release and binding of calcium in intracellular pools. Since they are inducers of vascular and other smooth muscle relaxation, they are used in the drug therapy of hypertension and cerebrovascular spasms, as myocardial protective agents, and in the relaxation of uterine spasms.  vasodilators; D25-26 qualif; DF: CA CHANNEL BLOCK   
See Also Antihypertensive Agents; Vasodilator Agents; Anti-Arrhythmia Agents
Other names Channel Blockers, Calcium; Calcium Inhibitors, Exogenous; Calcium Blockaders, Exogenous; Calcium Antagonists, Exogenous; Inhibitors, Exogenous Calcium; Blockers, Calcium Channel; Blockaders, Exogenous Calcium; Antagonists, Exogenous Calcium; Exogenous Calcium Inhibitors; Exogenous Calcium Blockaders; Exogenous Calcium Antagonists; Calcium Channel Blocking Drugs; Channel Blockers, Calcium; Calcium Inhibitors, Exogenous; Calcium Blockaders, Exogenous; Calcium Antagonists, Exogenous
Substances having this pharmacologic action: Lidoflazine; Bencyclane; carboxyamido-triazole; dotarizine; Nifedipine; TMB 8; Felodipine; Bepridil; Flunarizine; 1,4-dihydropyridine; gabapentin; falipamil; eperisone; PN 202-791; mepirodipine; KW 3049; KT 362; fenamic acid; azimilide; 1-(2-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenylethyl)-1H-imidazole; sesamodil; naftopidil; KB 2796; emopamil; AE0047; Conus magus toxin; piperidine; niludipin; 2-(4-(dimethylamino)styryl)-1-methylpyridinium; oxodipine; niguldipine; CD 349; enpiperate; Cinnarizine; cilnidipine; efonidipine; Verapamil; monatepil; Nisoldipine; Nimodipine; Nitrendipine; N-(2-guanidinoethyl)-5-isoquinolinesulfonamide; bevantolol; tranilast; nimesulide; Isradipine; Amlodipine; manidipine; R 56865; Perhexiline; Win 55212-2; Prenylamine; anipamil; pinaverium; devapamil; Mibefradil; clentiazem; ochratoxin A; FTX, spider toxin; octylonium; vinpocetine; dimeditiapramine; tetrahydropalmatine; risedronic acid; Magnesium Sulfate; omega-Conotoxin GVIA; omega-Agatoxin IVA; Conotoxins; omega-Conotoxins; manoalide; Gallopamil; SAN 202791; ryodipine; tetrandrine; tolfenamic acid; Amrinone; osthol; norverapamil; omega-conotoxin-MVIIC; fantofarone; NS 21; Diltiazem; ziconotide; lacidipine; lercanidipine; Nicardipine; darodipine; anandamide; IH 764-3; benidipine; lamotrigine; pranidipine; nilvadipine; berbamine; canadine; dauricine; fosfedil; Salvia miltiorrhizae extract; fasudil; stepholidine; terodiline; Fendiline; tetramethylpyrazine
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
propiverine  60569-19-9   *Benzilates Antiparkinson Agents Calcium Channel Blockers Urinary Incontinence. 
Pharma Action Parasympatholytics ; Cholinergic Antagonists
Psychiat Neurol Med Psychol 20(21):77;1975
azelnidipine  123524-52-7 3,5-Pyridinedicarboxylic acid, 2-amino-1,4-dihydro-6-methyl-4-(3-nitrophenyl)-, 3-(1-(diphenylmethyl)-3-azetidinyl) 5-(1-methylethyl) ester, (+- *Dihydropyridines Azetidinecarboxylic Acid/*analogs & derivatives Calcium Channel Blockers.  Jpn J Pharmacol 1989;51(1):57
ryosidine  89964-00-1   Organic Chemicals Calcium Channel Blockers.  Naunyn Schmiedebergs Arch Pharmacol 1984;325(2):124
AWD 160-275  0   *Amino Acids *Cyclohexylamines Calcium Channel Blockers.  Vestn Ross Akad Med Nauk 1998;(11):42-6
PD 173212  0   *Dipeptides Calcium Channel Blockers.  Bioorg Med Chem Lett 1999 Jul 5;9(13):1813-8
R 33956  87495-26-9 R 33956  Organic Chemicals Calcium Channel Blockers.  Am J Physiol 1983;244(3):C150
falicor  0   Organic Chemicals Calcium Channel Blockers.  Klin Med (Mosk) 1990;68(10):83
OF 5015  0   Organic Chemicals Calcium Channel Blockers.  Biull Eksp Biol Med 1993 Sep;116(9):288-90