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Cholinergic Antagonists
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Definition
: Drugs that bind to but do not activate CHOLINERGIC RECEPTORS, thereby blocking the actions of ACETYLCHOLINE or cholinergic agonists.
DF: CHOLINERGIC ANTAG
Examples
Muscarinic Antagonists
;
Nicotinic Antagonists
Other names
Cholinergic Blocking Agents; Anti Cholinergics; Antagonists, Cholinergic; Antagonists, Acetylcholine; Antagonist, Cholinergic; Agents, Cholinergic-
Blocking; Agents, Anticholinergic; Cholinergic Antagonist; Anticholinergics; Anti-
Cholinergics; Cholinergic-
Blocking Agents; Anticholinergic Agents; Cholinolytics; Acetylcholine Antagonists
Substances having this pharmacologic action:
Ipratropium
;
Scopolamine Hydrobromide
;
propiverine
;
desloratadine
;
NS 21
;
tiotropium
Substance
CAS Registry & name
Categories
Source
Drugs
*
atractylenolide I
0
*Lactones
*Sesquiterpenes
Cholinergic Antagonists.
Acta Pharmacol Sin 2000 Jan;21(1):91-6
4,15-
epoxy-
8-
hydroxyasterolide
0
*Lactones
*Sesquiterpenes
Cholinergic Antagonists.
Acta Pharmacol Sin 2000 Jan;21(1):91-6
atractylenolide III
0
*Lactones
*Sesquiterpenes
Cholinergic Antagonists.
Acta Pharmacol Sin 2000 Jan;21(1):91-6