encyclopedia of medical concepts
ψ
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Purinergic P1 Receptor Antagonists
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Definition
: Compounds that bind to and block the stimulation of PURINERGIC P1 RECEPTORS.
Examples
Adenosine A1 Receptor Antagonists
;
Adenosine A2 Receptor Antagonists
;
Adenosine A3 Receptor Antagonists
Other names
Receptor Antagonists, Adenosine; Purinoceptor Antagonists, P1; Antagonists, P1 Purinoceptor; Antagonists, Adenosine Receptor; P1 Purinoceptor Antagonists; Adenosine Receptor Antagonists
Substances having this pharmacologic action:
8-(4-sulfophenyl)theophylline
;
Theophylline
;
Caffeine
;
Aminophylline
;
1,3-dipropyl-8-(4-sulfophenyl)xanthine
;
8-cyclopentyl-1,3-dimethylxanthine
Substance
CAS Registry & name
Categories
Source
Drugs
*
2-
amino-
4-
phenyl-
8-
pyrrolidin-
1-
ylmethylindeno(1,2-
d)pyrimidin-
5-
one
0
*Indenes
*Pyrimidines
Receptor, Adenosine A1
Receptor, Adenosine A2A
Purinergic P1 Receptor Antagonists.
Chem Res Toxicol 2011 Jul 18;24(7):1012-30
4-
allyl-
8-
ethyl-
7,8-
dihydro-
2-
(3-
methoxy-
1-
methyl-
1H-
pyrazol-
5-
yl)-
1H-
imidazo(2,1-
i)purin-
5(4H)-
one
0
*Purines
Receptor, Adenosine A3
Purinergic P1 Receptor Antagonists.
J Med Chem 2011 Jul 28;54(14):5205-20