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Receptors, CXCR4
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Definition
: CXCR receptors with specificity for CXCL12 CHEMOKINE. The receptors may play a role in HEMATOPOIESIS regulation and can also function as coreceptors for the HUMAN IMMUNODEFICIENCY VIRUS.
DF: RECEPT CXCR4
Other names
Receptor, CXCR4; Leukocyte Derived Seven Transmembrane Domain Recep; Receptor, LESTR; Leukocyte-
Derived Seven-
Transmembrane Domain Recep; LESTR Receptor; CXCR4 Receptor; Fusin; CXCR4 Receptors; CXC Chemokine Receptor 4
Substance
CAS Registry & name
Categories
Source
Drugs
*
AMD 11070
0
*Aminoquinolines
*Benzimidazoles
Receptors, CXCR4/antagonists & inhibitors.
Mol Pharmacol 2008 Dec;74(6):1485-95
CXCR4a protein, zebrafish
0
*Receptors, CXCR4
*Zebrafish Proteins.
Science 2008 Oct 3;322(5898):89-92
CXCR4 protein, human
0
*Receptors, CXCR4.
J Immunol 1999 Sep 1;163(5):2368-72
N,N'-
di-
2-
pyridinyl-
1,4-
benzenedimethanamine
0
*Aminopyridines
*Benzylamines
Receptors, CXCR4/antagonists & inhibitors.
J Med Chem 2007 Nov 15;50(23):5655-64
1-
pyridin-
2-
yl-
N-
(4-
(1,4,7-
triazacyclotetradecan-
4-
ylmethyl)benzyl)methanamine
0
*Pyridines
Receptors, CXCR4/antagonists & inhibitors.
FASEB J 2007 Oct;21(12):3219-30
cyclo(tyrosyl-
methylarginyl-
arginyl-
3-
(2-
naphthyl)alanyl-
glycyl)
0
*Peptides, Cyclic
Receptors, CXCR4/antagonists & inhibitors.
J Med Chem 2007 Jan 25;50(2):192-8
cyclo(tyrosyl-
arginyl-
arginyl-
3-
(2-
naphthyl)alanyl-
alanyl)
0
*Peptides, Cyclic
Receptors, CXCR4/antagonists & inhibitors.
J Med Chem 2007 Jan 25;50(2):192-8
POL2438 peptide
0
*Peptides, Cyclic
Receptors, CXCR4/antagonists & inhibitors.
Bioorg Med Chem 2006 Dec 15;14(24):8396-404
T22 peptide
0
*Peptides
Receptors, CXCR4/antagonists & inhibitors.
Mol Cancer Ther 2006 Oct;5(10):2592-9
5,5'-
(1,4-
phenylenebis(methylene))bis(1,5,8,12-
tetraazabicyclo(10.2.2)hexadecane)
0
*Bicyclo Compounds, Heterocyclic
Receptors, CXCR4/antagonists & inhibitors.
J Med Chem 2006 Oct 19;49(21):6162-5
CXCR4 protein, mouse
0
*Receptors, CXCR4.
J Biol Chem 2006 Sep 22;281(38):27765-72
N-
(1,4,8,11-
tetraazacyclotetradecanyl-
1,4-
phenylenebis(methylene))-
2-
(aminomethyl)-
pyridine
0
*Pyridines
Receptors, CXCR4/antagonists & inhibitors.
Biochem Pharmacol 2005 Sep 1;70(5):752-61
cyclo(tyrosyl-
arginyl-
arginyl-
3-
(2-
naphthyl)alanyl-
glycyl)
0
*Peptides, Cyclic
Receptors, CXCR4/antagonists & inhibitors.
J Med Chem 2005 Jan 27;48(2):380-91
Cxcr4 protein, rat
0
*Receptors, CXCR4.
KRH 1636
0
*Pyridines
Arginine/*analogs & derivatives
Receptors, CXCR4/antagonists & inhibitors.
Proc Natl Acad Sci U S A 2003 Apr 1;100(7):4185-90
odysseus protein, zebrafish
0
*Receptors, CXCR4
*Zebrafish Proteins.
Nature 2003 Jan 16;421(6920):279-82
CGA 137053
0
*Amides
*Imidazoles
Receptors, CXCR4/antagonists & inhibitors.
Chem Biol 2000 Sep;7(9):669-76
TW 70
0
*Peptides, Cyclic
Receptors, CXCR4/antagonists & inhibitors.
Bioorg Med Chem 1998 Feb;6(2):231-8
JM 3100
155148-31-5
*Heterocyclic Compounds
Receptors, CXCR4/antagonists & inhibitors
HIV Fusion Inhibitors.
Pharma Action
Anti-HIV Agents
Antimicrob Agents Chemother 1994 Apr;38(4):668-74
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