encyclopedia of medical concepts
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Adrenergic alpha-1 Receptor Antagonists
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Definition
: Drugs that bind to and block the activation of ADRENERGIC ALPHA-1 RECEPTORS.
Other names
alpha1-
Antagonists, Adrenergic; alpha1 Adrenoceptor Blocker; alpha-
1 Antagonists, Adrenergic; alpha 1 Adrenergic Blocking Agents; Adrenergic alpha1 Antagonists; Adrenergic alpha 1 Receptor Blockers; Adrenergic alpha 1 Receptor Antagonists; alpha1-
Adrenoceptor Blocker; alpha-
1 Adrenergic Blocking Agents; Adrenergic alpha 1 Antagonists; Adrenergic alpha1-
Antagonists; Adrenergic alpha-
1 Receptor Blockers; Adrenergic alpha-
1 Antagonists
Substances having this pharmacologic action:
bunazosin
;
bucindolol
;
trimazosin
;
Terazosin
;
Labetalol
;
Prazosin
;
Doxazosin
;
Indoramin
;
urapidil
;
tamsulosin
;
carvedilol
;
alfuzosin
Substance
CAS Registry & name
Categories
Source
Drugs
*
3-
(4-
(ethylthio)-
1H-
benzimidazol-
2-
yl)isoquinoline
0
*Benzimidazoles
*Isoquinolines
Adrenergic alpha-1 Receptor Antagonists.
ChemMedChem. 2011 Oct 4;6(10):1909-18.
7-
(2-
hydroxypropoxy)-
3,4-
dihydroisoquinolin-
1(2H)-
one
0
*Isoquinolines
Adrenergic alpha-1 Receptor Antagonists.
Chem Biol Drug Des. 2010 Dec;76(6):505-10