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ψ
GABA Agonists
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Definition
: Endogenous compounds and drugs that bind to and activate GAMMA-AMINOBUTYRIC ACID receptors (RECEPTORS, GABA).
note specifics; do not confuse with GABA ANTAGONISTS
Examples
GABA-A Receptor Agonists
;
GABA-B Receptor Agonists
Other names
gamma Aminobutyric Acid Agonists; gamma Aminobutyric Acid Agonist; Receptor Agonists, GABA; Receptor Agonist, GABA; Agonists, gamma-
Aminobutyric Acid; Agonists, GABA Receptor; Agonists, GABA; Agonist, gamma-
Aminobutyric Acid; Agonist, GABA Receptor; Agonist, GABA; Acid Agonists, gamma-
Aminobutyric; Acid Agonist, gamma-
Aminobutyric; gamma-
Aminobutyric Acid Agonist; GABA Receptor Agonists; GABA Receptor Agonist; GABA Agonist; gamma-
Aminobutyric Acid Agonists
Substances having this pharmacologic action:
progabide
;
piperidine-4-sulfonic acid
;
2-phenylpyrazolo(4,3-c)quinolin-3(5H)-one
;
4-amino-3-phenylbutyric acid
;
homotaurine
;
isoguvacine
;
4,5,6,7-tetrahydroisoxazolo(5,4-c)pyridin-3-ol
;
3-aminopropylphosphinic acid
;
tiagabine
Substance
CAS Registry & name
Categories
Source
Drugs
*
7-
((2-
(3-
fluoropyridin-
2-
yl)-
1H-
imidazol-
1-
yl)methyl)-
2-
methyl-
8-
propyl-
(1,2,4)triazolo(1,5-
c)pyrimidine
0
*Pyrimidines
*Triazoles
Receptors, GABA-A
GABA Agonists.
Eur J Pharmacol. 2011 Oct 1;668(1-2):190-3.