encyclopedia of medical concepts
ψ
ψ
Purinergic P2Y Receptor Antagonists
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Definition
: Compounds that bind to and block the stimulation of PURINERGIC P2Y RECEPTORS. Included under this heading are antagonists for specific P2Y receptor subtypes.
Other names
P2Y1 Purinoceptor Antagonists; ADP Receptor Blockers; ADP Receptor Antagonists; Receptor Blockers, ADP; Receptor Antagonists, ADP; Purinoceptor Antagonists, P2Y2; Purinoceptor Antagonists, P2Y12; Purinoceptor Antagonists, P2Y1; Purinoceptor Antagonists, P2Y; Blockers, ADP Receptor; Antagonists, P2Y2 Purinoceptor; Antagonists, P2Y12 Purinoceptor; Antagonists, P2Y1 Purinoceptor; Antagonists, P2Y Purinoceptor; Antagonists, ADP Receptor; Purinergic P2Y2 Receptor Antagonists; Purinergic P2Y12 Receptor Antagonists; Purinergic P2Y1 Receptor Antagonists; P2Y2 Purinoceptor Antagonists; P2Y12 Purinoceptor Antagonists
Substances having this pharmacologic action:
Ticlopidine
;
N(6)-methyl-2'-deoxyadenosine 3',5'-diphosphate
;
cangrelor
;
prasugrel
;
Ticagrelor
;
clopidogrel
Substance
CAS Registry & name
Categories
Source
Drugs
*
2-
chloro-
N6-
methyl-
(N)-
methanocarba-
2'-
deoxyadenosine-
3',5'-
bisphosphate
0
Adenosine Diphosphate/*analogs & derivatives
Purinergic P2Y Receptor Antagonists.
Br J Pharmacol 2002 Apr;135(8):2004-10