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Flumazenil
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Definition
: A potent benzodiazepine receptor antagonist. Since it reverses the sedative and other actions of benzodiazepines, it has been suggested as an antidote to benzodiazepine overdoses.
Pharmacological Action
Antidotes
;
GABA Modulators
Other names
Flumazepil; Ro 151788; Ro 15 1788; Hoffman La Roche Brand of Flumazenil; Romazicon; Roche Brand of Flumazenil; Ro 15-
1788; Lanexat; Hoffman-
La Roche Brand of Flumazenil; Anexate
Drugs
*
:
FLUMAZENIL
;
ROMAZICON
Substance
CAS Registry & name
Categories
Source
Drugs
*
2'-
fluoroflumazenil
0
Flumazenil/*analogs & derivatives
Fluorine Radioisotopes.
Nucl Med Biol 2003 Jul;30(5):521-7
5-
(2'-
fluoroethylflumazenil)
0
Flumazenil/*analogs & derivatives.
Nucl Med Biol 2001 Oct;28(7):809-14
3-
(5-
cyclopropyl-
1,2,4-
oxadiazol-
3-
yl) 7-
bromo-
5,6-
dihydro-
5-
methyl-
6-
oxo-
4H-
imidazo(1,5.alpha)-
benzodiazepine
0
*Oxadiazoles
Flumazenil
Receptors, GABA-A/agonists.
Eur J Nucl Med 1997 Oct;24(10):1261-7
5-
(2'-
fluoroethyl)flumazenil
143693-57-6
Flumazenil/*analogs & derivatives
Fluorine Radioisotopes.
Eur J Pharmacol 1992 Jul 21;218(1):109-15
ethyl 8-
fluoro-
5,6-
dihydro-
5-
(3'-
fluoropropyl)-
6-
oxo-
4H-
imidazol(1,5-
a)(1,4)benzodiazepine-
3-
carboxylate
133368-71-5
Flumazenil/*analogs & derivatives.
Int J Rad Appl Instrum (B) 1990;17(8):811
3'-
fluoropropyl-
8-
fluoro-
5,6-
dihydro-
5-
methyl-
6-
oxo-
4H-
imidazol(1,5-
a)(1,4)benzodiazepine-
3-
carboxylic acid
133368-73-7
Flumazenil/*analogs & derivatives.
Int J Rad Appl Instrum (B) 1990;17(8):811
BD 623
132305-66-9 4H-
Imidazo(1,5-
a)(1,4)benzodiazepine-
3-
carboxylic acid, 8-
fluoro-
5,6-
dihydro-
5-
methyl-
6-
oxo-
, 3-
((7-
nitro-
4-
benzofurazanyl)amino)propyl ester
Flumazenil/*analogs & derivatives
4-Chloro-7-nitrobenzofurazan/*analogs & derivatives.
J Biol Chem 1990;265(36):22181
iomazenil
127396-36-5
Flumazenil/*analogs & derivatives
Iodine Radioisotopes.
Int J Rad Appl Instrum (B) 1989;16(8):759
Ro 15-
3890
84378-44-9
Flumazenil/*analogs & derivatives.
Int J Rad Appl Instrum (A) 1988;39(9):993