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Boronic Acids 
Inorganic or organic compounds that contain the basic structure RB(OH)2.  do not confuse with BORINIC ACIDS    Other names Acids, Boronic
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
bortezomib  0   *Boronic Acids *Pyrazines. 
Pharma Action Antineoplastic Agents ; Protease Inhibitors 		Clin Cancer Res 1999 Sep;5(9):2638-45VELCADE
benzeneboronic acid  98-80-6   *Boronic Acids.  Biochim Biophys Acta 525(2):423;1978; J Bacteriol 136(2):625;1978; J Biochem (Tokyo) 77(4):905;1975; J Biochem (Tokyo) 79(1):107;1976; J Biochem (Tokyo) 80:491;1976; J Biochem (Tokyo) 81:1269;1977
3-aminobenzeneboronic acid  30418-59-8   *Boronic Acids.  J Bacteriol 1981;145(1):489
MG 262  0   *Boronic Acids.  Proc Natl Acad Sci U S A 2001 Jan 16;98(2):513-8
3-nitrobenzeneboronic acid  13331-27-6   *Boronic Acids.  Biochim Biophys Acta 524(2):413;1978
methyl-O-succinyl-alanyl-alanyl-prolyl-borovaline-pinacol  94242-92-9   *Boronic Acids *Oligopeptides Pancreatic Elastase Pancreatic Elastase/antagonists & inhibitors.  Am Rec Respir Dis 1986;133(4):635
benzo(b)thiophene-2-boronic acid  0   *Boronic Acids *Thiophenes beta-Lactamases/antagonists & inhibitors beta-Lactam Resistance.  J Med Chem 1998 Nov 5;41(23):4577-86
N-dansyl-3-aminobenzeneboronic acid  75806-94-9 Boronic acid, (3-(((5-(dimethylamino)-1-naphthalenyl)sulfonyl)amino)phenyl)  *Boronic Acids *Dansyl Compounds Subtilisins/antagonists & inhibitors.  Biochem Biophys Res Commun 1980;96(1):157; FEBS Lett 1981;133(1):36
(2-boronoethyl)-cysteine  0   Arginase/antagonists & inhibitors *Boronic Acids.  Biochemistry 2001 Mar 6;40(9):2678-88
PT-100 dipeptide  0   *Boronic Acids *Dipeptides.  Blood. 2003 Sep 1;102(5):1641-8
phenylethane boronic acid  34420-17-2 Boronic acid, (2-phenylethyl)  *Boronic Acids.  J Biol Chem 1983;258(4):2135
dihydroxyboronyl-sepharose  125022-86-8   *Boronic Acids *Sepharose.  Anal Biochem 1988;174(1):239
3-acrylamidophenylboronic acid  0   *Boronic Acids.  Biotechnol Bioeng 2001 Feb 5;72(3):307-14
1-acetamido-2-(4-fluorophenyl)ethane-1-boronic acid  149982-17-2   *Boronic Acids *Fluorobenzenes.  Biochim Biophys Acta 1993 Jun 4;1163(3):321-34
O-methyl-succinyl-alanyl-alanyl-prolyl-borovaline  94242-73-6   *Boronic Acids *Oligopeptides.  Biochemistry 1993 Nov 30;32(47):12651-5
3-propionamidophenylboronic acid  153853-43-1   *Boronic Acids.  J Biochem (Tokyo) 1995 Jun;117(6):1145-7
phenylborate polymer  0   *Boronic Acids *Polymers.  Pharm Res 1997 Mar;14(3):289-93
N-tert-butyloxycarbonyl-Ala-Pro-boroVal  0   *Boronic Acids *Oligopeptides.  J Biomol NMR 1997 Jul;10(1):21-7
4-vinylphenyl boronic acid  0   *Boronic Acids *Vinyl Compounds.  J Biomater Sci Polym Ed 2000;11(8):817-31
Phe-Leu boronic acid  0   *Boronic Acids *Dipeptides.  Transplantation 2001 Jul 27;72(2):196-202
4-(4,5-diphenyl-1H-imidazol-2-yl)phenylboronic acid  0   *Boronic Acids *Imidazoles.  J Chromatogr A. 2005 Feb 25;1066(1-2):119-25
3,5-bis(4-boronic acid-benzylidene)-1-methylpiperidin-4-one  0   *Boronic Acids *Piperidines.  Bioorg Med Chem 2006 May 15;14(10):3491-5
N,N'-bis(3-(dihydroxylborylbenzene))adipamide  75806-95-0 Boronic acid, ((1,6-dioxo-1,6-hexanediyl)bis(imino-3,1-phenylene))bis  *Boronic Acids.  Biochem Biophys Res Commun 1980;96(1):157
3-nitro-4-(6-aminohexylamido)phenylboronic acid  80500-29-4 Boronic acid, (4-(((6-aminohexyl)amino)carbonyl)-3-nitrophenyl)  *Boronic Acids.  Biochem J 1981;197(3):683
4-carboxy-2-nitrobenzeneboronic acid  85107-54-6   *Boronic Acids.  Acta Crystallogr C 1993 Apr 15;49(Pt 4):690-3
poly(AAm-co-PBA)  0   *Acrylic Resins *Boronic Acids.  Biochem Biophys Res Commun 1993 Sep 15;195(2):829-36
O-methylsuccinyl-alanyl-alanyl-prolyl-borophenylalanine  97590-10-8   *Boronic Acids *Oligopeptides.  Biochemistry 1993 Nov 30;32(47):12651-5
3-methacrylamidophenylboronic acid  48150-45-4   *Boronic Acids *Methacrylates.  Biomaterials 1994 Jan;15(2):121-8
1-acetamido-2-(3-carboxyphenyl)ethane boronic acid  0   *Acetamides *Boronic Acids.  Nat Struct Biol 1996 Aug;3(8):688-95
1,1'-biphenyl-4-yl-boronic acid  5122-94-1   *Boronic Acids.  J Biolumin Chemilumin 1996 May-Jun;11(3):137-47
alanylpyrrolidine-boronic acid  0   *Dipeptides Boronic Acids.  Int J Immunopharmacol 1997 Jan;19(1):15-24
(1-acetamido-2-(4-chlorophenyl)ethyl)boronic acid  0   *Boronic Acids.  Biochemistry 1998 Jan 13;37(2):451-62
(1-acetamido-2-(1-naphthyl)ethyl)boronic acid  0   *Boronic Acids.  Biochemistry 1998 Jan 13;37(2):451-62
PS 273  0   *Boronic Acids *Dipeptides.  Methods Enzymol 1999;300:345-63
4-boronic acid benzophenone  0   Subtilisin/antagonists & inhibitors *Benzophenones *Boronic Acids.  Bioorg Med Chem 2000 Mar;8(3):563-70
diisopropyl 2-bora-2-(3-(phenyldimethylsilyl)-2-propen-1-yl)-1,3-dioxole-4,5-dicarboxylate  0   *Boronic Acids *Organosilicon Compounds.  Org Lett 2000 Feb 24;2(4):461-4
1-phenylacetamido-2-(3-carboxyphenyl)ethylboronic acid  0   *Boronic Acids.  Biochemistry 2000 May 9;39(18):5312-21
1-acetamido-2-(3-carboxy-2-hydroxyphenyl)ethylboronic acid  0   *Boronic Acids.  Biochemistry 2000 May 9;39(18):5312-21
1-aminocyclopropaneboronic acid  0   Protease Inhibitors *Boronic Acids *Cyclopropanes.  Org Lett 2000 Oct 5;2(20):3095-7
4-(4,5-di(2-pyridyl)-1H-imidazol-2-yl)phenylboronic acid  0   *Boronic Acids.  Luminescence 2001 Mar-Apr;16(2):167-72
tolylboronic acid  0   *Boronic Acids.  Org Lett 2001 Jun 28;3(13):2077-9
glutamyl-gamma-boronate  0   Glutamates *Boronic Acids.  Bioorg Med Chem Lett 2001 Sep 17;11(18):2561-4
4'-cyanostilbene-4-boronic acid  0   Fluorescent Dyes *Boronic Acids *Stilbenes.  Anal Biochem 2002 Feb 1;301(1):111-6
alanyl-boroalanine  0   *Boronic Acids *Dipeptides.  Adv Exp Med Biol 2003;524:333-8
thianaphthene-2-boronic acid  0   *Boronic Acids *Thiophenes.  J Med Chem 2003 Jul 31;46(16):3448-51
8-quinolineboronic acid  0   *Boronic Acids *Quinolines.  Bioorg Med Chem Lett. 2003 Mar 24;13(6):1019-22
3-((1-((4-(5,6-dimethoxy-1-oxoisoindolin-2-yl)-2-methoxyphenyl)sulfonyl)pyrrolidin-2-yl)carbonylamino)phenylboronic acid  0   *Boronic Acids *Pyrrolidines.  J Chromatogr B Analyt Technol Biomed Life Sci. 2003 May 25;788(2):401-5
4-(dimethylamino)naphthalene-1-boronic acid  0   *Boronic Acids 1-Naphthylamine/*analogs & derivatives.  Org Lett 2003 Nov 27;5(24):4599-602
dansyl-3-aminophenylboronate  0   *Boronic Acids *Dansyl Compounds.  Rapid Commun Mass Spectrom. 2004;18(7):816-21
2-methylphenyl boronic acid  0   *Boronic Acids.  Angew Chem Int Ed Engl. 2004 Mar 26;43(14):1871-6
4-amino-3-fluorophenylboronic acid  0   *Boronic Acids.  Clin Chem 2004 Dec;50(12):2353-60
4-carboxy-3-fluorophenylboronic acid  0   *Boronic Acids.  Clin Chem 2004 Dec;50(12):2353-60
thiolate boronic acid  0   *Boronic Acids *Sulfhydryl Compounds.  Anal Biochem 2004 Sep 15;332(2):253-60
N-(o-boronic acid)benzyl-1-naphthylamine  0   *Boronic Acids 1-Naphthylamine/*analogs & derivatives.  Luminescence 2005 Jul-Oct;20(4-5):331-3
3-(4-(3-phenyl-2-pyrazolin-1-yl)benzene-1-sulfonylamido)phenylboronic acid  0   Myosins/antagonists & inhibitors *Boronic Acids *Sulfonamides.  Biochemistry 2006 Jan 31;45(4):1234-41
N-(4-morpholine)carbonyl-beta-(1-naphthyl)-alanyl-leucine boronic acid  0   *Boronic Acids *Dipeptides.  Mol Microbiol 2006 Mar;59(5):1417-28
4-mercaptophenylboronic acid  0   *Boronic Acids *Sulfhydryl Compounds.  Langmuir. 2005 May 24;21(11):5101-7
dithiobis(4-butyrylamino-m-phenylboronic acid)  0   *Boronic Acids *Sulfhydryl Compounds.  Langmuir. 2005 May 24;21(11):5101-7
polyvinylamine-poly(4-carboxyphenylboronic acid)  0   *Boronic Acids *Polyvinyls.  Biomacromolecules 2006 Mar;7(3):701-2
beta-(4-borono-2,6-difluorophenyl)alanine  0   *Boronic Acids Phenylalanine/*analogs & derivatives.  Bioorg Med Chem 2006 May 15;14(10):3258-62
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