encyclopedia of medical concepts
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AG 127
under Tyrphostins
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Tyrphostins
Definition
: A family of synthetic protein tyrosine kinase inhibitors. They selectively inhibit receptor autophosphorylation and are used to study receptor function.
Substance
CAS Registry & name
Categories
Source
Drugs
*
AG 127 [ AG 126,AG-126,AG-127,AG126,alpha-cyano-(3-hydroxy-4-nitro)cinnamonitrile,tyrphostin AG127 ]
structure given in first source
118409-62-4
*Tyrphostins
Protein-Tyrosine Kinases/antagonists & inhibitors
Pharma Action
Enzyme Inhibitors
Biochem Biophys Res Commun 1991;176(3):1425